CPIC Guidelines Only (103 Drugs) CPIC Guidelines and FDA Table (50 Drugs)* FDA Table Only (64 Drugs)
  1. Aceclofenac
  2. Alfentanil
  3. Amikacin
  4. Aminosalicylic acid
  5. Aspirin
  6. Atazanavir
  7. Buprenorphine
  8. Chloramphenicol
  9. Chloroquine
  10. Chlorpropamide
  11. Ciprofloxacin
  12. Dabrafenib
  13. Dapsone
  14. Desflurane
  15. Desvenlafaxine
  16. Dibekacin
  17. Diclofenac
  18. Dimercaprol
  19. Doxorubicin
  20. Duloxetine
  21. Enflurane
  22. Fentanyl
  23. Fluoxetine
  24. Fluvastatin
  25. Furazolidone
  26. Gentamicin
  27. Gliclazide
  28. Glimepiride
  29. Glipizide
  30. Glyburide
  31. Halothane
  32. Hydrocodone
  33. Hydromorphone
  34. Hydroxychloroquine
  35. Indomethacin
  36. Isoflurane
  37. Ivacaftor
  38. Kanamycin
  39. Levomethadone
  40. Levomilnacipran
  41. Lornoxicam
  42. Lovastatin
  43. Lumiracoxib
  44. Mafenide
  45. Mepacrine
  46. Mesalazine
  47. Metamizole
  48. Methadone
  49. Methoxyflurane
  50. Methylene blue
  51. Milnacipran
  52. Morphine
  53. Moxifloxacin
  54. Nabumetone
  55. Nalidixic acid
  56. Naltrexone
  57. Naproxen
  58. Neomycin
  59. Netilmicin
  60. Nicorandil
  61. Nitrofural
  62. Nitrofurantoin
  63. Norfloxacin
  64. Ofloxacin
  65. Ondansetron
  66. Oxycodone
  67. Paromomycin
  68. Peginterferon alfa-2a
  69. Peginterferon alfa-2b
  70. Pegloticase
  71. Phenazopyridine
  72. Pitavastatin
  73. Plazomicin
  74. Pravastatin
  75. Primaquine
  76. Probenecid
  77. Quinine
  78. Rasburicase
  79. Remifentanil
  80. Ribavirin
  81. Ribostamycin
  82. Sertraline
  83. Sevoflurane
  84. Sodium nitrite
  85. Streptomycin
  86. Sufentanil
  87. Sulfacetamide
  88. Sulfadiazine
  89. Sulfadimidine
  90. Sulfanilamide
  91. Sulfisoxazole
  92. Tafenoquine
  93. Tegafur
  94. Tenoxicam
  95. Tobramycin
  96. Tolazamide
  97. Tolbutamide
  98. Toluidine blue
  99. Trametinib
  100. Tropisetron
  101. Vilazodone
  102. Vitamin C
  103. Vitamin K
  1. Abacavir
  2. Allopurinol
  3. Amitriptyline
  4. Atomoxetine
  5. Atorvastatin
  6. Azathioprine
  7. Capecitabine
  8. Carbamazepine **
  9. Celecoxib
  10. Citalopram
  11. Clomipramine
  12. Clopidogrel
  13. Codeine **
  14. Desipramine
  15. Dexlansoprazole
  16. Doxepin
  17. Efavirenz
  18. Escitalopram
  19. Esomeprazole
  20. Fluorouracil
  21. Flurbiprofen
  22. Fluvoxamine
  23. Fosphenytoin
  24. Ibuprofen
  25. Imipramine
  26. Lansoprazole
  27. Meloxicam
  28. Mercaptopurine
  29. Nortriptyline
  30. Omeprazole
  31. Oxcarbazepine
  32. Pantoprazole
  33. Paroxetine
  34. Phenytoin
  35. Piroxicam
  36. Rabeprazole
  37. Rosuvastatin
  38. Simvastatin
  39. Succinylcholine
  40. Sulfamethoxazole/Trimethoprim
  41. Sulfasalazine
  42. Tacrolimus
  43. Tamoxifen
  44. Thioguanine
  45. Tramadol **
  46. Trimipramine
  47. Venlafaxine
  48. Voriconazole
  49. Vortioxetine
  50. Warfarin
  1. Abrocitinib
  2. Amifampridine
  3. Amifampridine phosphate
  4. Amoxapine
  5. Amphetamine
  6. Aripiprazole
  7. Aripiprazole lauroxil
  8. Avatrombopag
  9. Belinostat
  10. Belzutifan
  11. Brexpiprazole
  12. Brivaracetam
  13. Carisoprodol
  14. Carvedilol
  15. Cevimeline
  16. Clobazam
  17. Clozapine
  18. Darifenacin
  19. Deutetrabenazine
  20. Diazepam
  21. Dolutegravir
  22. Donepezil
  23. Dronabinol
  24. Elagolix
  25. Eliglustat
  26. Erdafitinib
  27. Fesoterodine
  28. Flibanserin
  29. Galantamine
  30. Gefitinib
  31. Hydralazine
  32. Iloperidone
  33. Irinotecan
  34. Isoniazid
  35. Lapatinib
  36. Lofexidine
  37. Mavacamten
  38. Meclizine
  39. Metoclopramide
  40. Metoprolol
  41. Mirabegron
  42. Mivacurium
  43. Nateglinide
  44. Nebivolol
  45. Nilotinib
  46. Oliceridine
  47. Pazopanib
  48. Perphenazine
  49. Pimozide
  50. Pitolisant
  51. Procainamide
  52. Propafenone
  53. Propranolol
  54. Protriptyline
  55. Raltegravir
  56. Risperidone
  57. Sacituzumab
  58. Siponimod
  59. Tamsulosin
  60. Tetrabenazine
  61. Thioridazine
  62. Tolterodine
  63. Valbenazine
  64. Viloxazine

 

Abbreviations: CPIC (Clinical Pharmacogenetics Implementation Consortium); FDA (Food and Drug Administration); PK (pharmacokinetics).
* Reflects CPIC provisional levels.
** Carbamazepine, codeine, and tramadol are listed in two FDA sections for different gene-drug associations.